Synthesis and Fluorescence Properties of new Monastrol Analogs Conjugated Fluorescent Coumarin Scaffolds
| dc.contributor.author | Al-Masoudi, Najim A. | |
| dc.contributor.author | Al-Salihi, Niran J. | |
| dc.contributor.author | Marich, Yossra A. | |
| dc.contributor.author | Markus, Timo | |
| dc.date.accessioned | 2017-08-10T09:36:57Z | |
| dc.date.available | 2017-08-10T09:36:57Z | |
| dc.date.issued | 2016 | eng |
| dc.description.abstract | A mild and efficient method has been used for the synthesis of ethyl 4-(3-hydroxphenyl)-6-methyl-2-thioxo-1,3-dihydroprimidine-5-carboxylate (monastrol) (2), via Biginelli reaction. Alkylation of 2 with the fluorescent coumarin 3 afforded the new thioether analog 4. Similarly, ethyl 4-(6,8-dichloro-2-oxo-2 H-chromen-3-yl)-6-methyl-2-thioxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylate (6) was prepared. The synthesized compounds are fluorescent active and show wavelength of maximum absorption (λmax) in UV or visible region in MeOH at room temperature. | eng |
| dc.description.version | published | eng |
| dc.identifier.doi | 10.1007/s10895-015-1695-x | eng |
| dc.identifier.pmid | 26498456 | eng |
| dc.identifier.uri | https://kops.uni-konstanz.de/handle/123456789/39824 | |
| dc.language.iso | eng | eng |
| dc.subject.ddc | 540 | eng |
| dc.title | Synthesis and Fluorescence Properties of new Monastrol Analogs Conjugated Fluorescent Coumarin Scaffolds | eng |
| dc.type | JOURNAL_ARTICLE | eng |
| dspace.entity.type | Publication | |
| kops.citation.bibtex | @article{AlMasoudi2016Synth-39824,
year={2016},
doi={10.1007/s10895-015-1695-x},
title={Synthesis and Fluorescence Properties of new Monastrol Analogs Conjugated Fluorescent Coumarin Scaffolds},
number={1},
volume={26},
issn={1053-0509},
journal={Journal of Fluorescence},
pages={31--35},
author={Al-Masoudi, Najim A. and Al-Salihi, Niran J. and Marich, Yossra A. and Markus, Timo}
} | |
| kops.citation.iso690 | AL-MASOUDI, Najim A., Niran J. AL-SALIHI, Yossra A. MARICH, Timo MARKUS, 2016. Synthesis and Fluorescence Properties of new Monastrol Analogs Conjugated Fluorescent Coumarin Scaffolds. In: Journal of Fluorescence. 2016, 26(1), pp. 31-35. ISSN 1053-0509. eISSN 1573-4994. Available under: doi: 10.1007/s10895-015-1695-x | deu |
| kops.citation.iso690 | AL-MASOUDI, Najim A., Niran J. AL-SALIHI, Yossra A. MARICH, Timo MARKUS, 2016. Synthesis and Fluorescence Properties of new Monastrol Analogs Conjugated Fluorescent Coumarin Scaffolds. In: Journal of Fluorescence. 2016, 26(1), pp. 31-35. ISSN 1053-0509. eISSN 1573-4994. Available under: doi: 10.1007/s10895-015-1695-x | eng |
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| kops.sourcefield | Journal of Fluorescence. 2016, <b>26</b>(1), pp. 31-35. ISSN 1053-0509. eISSN 1573-4994. Available under: doi: 10.1007/s10895-015-1695-x | deu |
| kops.sourcefield.plain | Journal of Fluorescence. 2016, 26(1), pp. 31-35. ISSN 1053-0509. eISSN 1573-4994. Available under: doi: 10.1007/s10895-015-1695-x | deu |
| kops.sourcefield.plain | Journal of Fluorescence. 2016, 26(1), pp. 31-35. ISSN 1053-0509. eISSN 1573-4994. Available under: doi: 10.1007/s10895-015-1695-x | eng |
| source.bibliographicInfo.fromPage | 31 | eng |
| source.bibliographicInfo.issue | 1 | eng |
| source.bibliographicInfo.toPage | 35 | eng |
| source.bibliographicInfo.volume | 26 | eng |
| source.identifier.eissn | 1573-4994 | eng |
| source.identifier.issn | 1053-0509 | eng |
| source.periodicalTitle | Journal of Fluorescence | eng |