Publikation: Monastrol analogs : a synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening
Lade...
Dateien
Datum
2010
Autor:innen
Herausgeber:innen
ISSN der Zeitschrift
Electronic ISSN
ISBN
Bibliografische Daten
Verlag
Schriftenreihe
Auflagebezeichnung
URI (zitierfähiger Link)
DOI (zitierfähiger Link)
Internationale Patentnummer
Link zur Lizenz
Angaben zur Forschungsförderung
Projekt
Open Access-Veröffentlichung
Open Access Green
Sammlungen
Core Facility der Universität Konstanz
Titel in einer weiteren Sprache
Publikationstyp
Zeitschriftenartikel
Publikationsstatus
Published
Erschienen in
Bioorganic & Medicinal Chemistry Letters. 2010, 20(14), pp. 4073-4076. ISSN 0960-894X. eISSN 1464-3405. Available under: doi: 10.1016/j.bmcl.2010.05.085
Zusammenfassung
A synthesis of novel pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged pyrazolo-, tetrazolo-, benzimidazo-, and thiazolopyrimidines via Hantzsch- and Biginelli-like condensations has been developed. The ability of these compounds to inhibit Eg5 activity has been examined. The results indicate that synthetic manipulations in the monastrol thiourea moiety are inefficient.
Zusammenfassung in einer weiteren Sprache
Fachgebiet (DDC)
570 Biowissenschaften, Biologie
Schlagwörter
Biginelli reaction, Hantzsch reaction, Oxygen-bridged nitrogen heterocycles, Monastrol analogs
Konferenz
Rezension
undefined / . - undefined, undefined
Zitieren
ISO 690
SVETLIK, Jan, Lucia VEIZEROVÁ, Thomas U. MAYER, Mario CATARINELLA, 2010. Monastrol analogs : a synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening. In: Bioorganic & Medicinal Chemistry Letters. 2010, 20(14), pp. 4073-4076. ISSN 0960-894X. eISSN 1464-3405. Available under: doi: 10.1016/j.bmcl.2010.05.085BibTex
@article{Svetlik2010-07-15Monas-12548, year={2010}, doi={10.1016/j.bmcl.2010.05.085}, title={Monastrol analogs : a synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening}, number={14}, volume={20}, issn={0960-894X}, journal={Bioorganic & Medicinal Chemistry Letters}, pages={4073--4076}, author={Svetlik, Jan and Veizerová, Lucia and Mayer, Thomas U. and Catarinella, Mario} }
RDF
<rdf:RDF xmlns:dcterms="http://purl.org/dc/terms/" xmlns:dc="http://purl.org/dc/elements/1.1/" xmlns:rdf="http://www.w3.org/1999/02/22-rdf-syntax-ns#" xmlns:bibo="http://purl.org/ontology/bibo/" xmlns:dspace="http://digital-repositories.org/ontologies/dspace/0.1.0#" xmlns:foaf="http://xmlns.com/foaf/0.1/" xmlns:void="http://rdfs.org/ns/void#" xmlns:xsd="http://www.w3.org/2001/XMLSchema#" > <rdf:Description rdf:about="https://kops.uni-konstanz.de/server/rdf/resource/123456789/12548"> <dcterms:available rdf:datatype="http://www.w3.org/2001/XMLSchema#dateTime">2011-06-21T07:34:25Z</dcterms:available> <dc:rights>terms-of-use</dc:rights> <dcterms:bibliographicCitation>First publ. in: Bioorganic & Medicinal Chemistry Letters 20 (2010), 14, pp. 4073-4076</dcterms:bibliographicCitation> <dc:contributor>Catarinella, Mario</dc:contributor> <dc:contributor>Veizerová, Lucia</dc:contributor> <foaf:homepage rdf:resource="http://localhost:8080/"/> <dc:contributor>Svetlik, Jan</dc:contributor> <dc:contributor>Mayer, Thomas U.</dc:contributor> <bibo:uri rdf:resource="http://kops.uni-konstanz.de/handle/123456789/12548"/> <void:sparqlEndpoint rdf:resource="http://localhost/fuseki/dspace/sparql"/> <dcterms:abstract xml:lang="eng">A synthesis of novel pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged pyrazolo-, tetrazolo-, benzimidazo-, and thiazolopyrimidines via Hantzsch- and Biginelli-like condensations has been developed. The ability of these compounds to inhibit Eg5 activity has been examined. The results indicate that synthetic manipulations in the monastrol thiourea moiety are inefficient.</dcterms:abstract> <dcterms:rights rdf:resource="https://rightsstatements.org/page/InC/1.0/"/> <dc:language>eng</dc:language> <dspace:hasBitstream rdf:resource="https://kops.uni-konstanz.de/bitstream/123456789/12548/1/svetlik.pdf"/> <dcterms:hasPart rdf:resource="https://kops.uni-konstanz.de/bitstream/123456789/12548/1/svetlik.pdf"/> <dc:creator>Catarinella, Mario</dc:creator> <dc:creator>Svetlik, Jan</dc:creator> <dc:creator>Veizerová, Lucia</dc:creator> <dc:creator>Mayer, Thomas U.</dc:creator> <dcterms:issued>2010-07-15</dcterms:issued> <dspace:isPartOfCollection rdf:resource="https://kops.uni-konstanz.de/server/rdf/resource/123456789/28"/> <dc:date rdf:datatype="http://www.w3.org/2001/XMLSchema#dateTime">2011-06-21T07:34:25Z</dc:date> <dcterms:isPartOf rdf:resource="https://kops.uni-konstanz.de/server/rdf/resource/123456789/28"/> <dcterms:title>Monastrol analogs : a synthesis of pyrazolopyridine, benzopyranopyrazolopyridine, and oxygen-bridged azolopyrimidine derivatives and their biological screening</dcterms:title> </rdf:Description> </rdf:RDF>
Interner Vermerk
xmlui.Submission.submit.DescribeStep.inputForms.label.kops_note_fromSubmitter
Prüfungsdatum der Dissertation
Finanzierungsart
Kommentar zur Publikation
Allianzlizenz
Corresponding Authors der Uni Konstanz vorhanden
Internationale Co-Autor:innen
Universitätsbibliographie
Ja